Ion Channel Screens & Concentration Response Assays

Functional, validated Ion Channel cell-based assays for screening and profiling

ChanTest’s Ion Channel portfolio includes over 90 targets. Applications of the portfolio include our NEW Ion Channel Panels™ that provide functional, automated ion channel screens by therapeutic target for profiling and safety assessment. Check back regularly for an updated listing of available targets.

Target Family Validation
5-HT3A Ligand-gated MP, PX
ASIC1a Acid-Sensing PX, QP
ASIC2a Acid-Sensing PX, QP
ASIC3 Acid-Sensing PX, QP
BK (KCa1.1) Potassium, calcium-activated PX, QP, FLP
Cav1.1/β1/α2δ (SKM L-type) Calcium, voltage-gated  
Cav1.2/β2/α2δ (Cardiac L-type) Calcium, voltage-gated MP, PX, QP, IWQ
Cav2.1/β4/α2δ (P/Q-type) Calcium, voltage-gated PX, QP, IWQ
Cav2.2/β3/α2δ (N-type) Calcium, voltage-gated MP, PX, QP, IWQ
Cav3.2 (T-type) Calcium, voltage-gated PX, QP, IWQ
CFTR Chloride PX, QP, IWQ
CLC-1 Chloride PX, QP
CLC-2 Chloride PX, QP
ENaC Sodium, epithelial  
GABA-A (α1/β2/γ2) Ligand-gated PX, QP
GABA-A (α2/β2/γ2) Ligand-gated PX, QP, FLP
GABA-A (α3/β2/γ2) Ligand-gated  
GABA-A (α5/β2/γ2) Ligand-gated PX, QP, FLP
HCN1 Hyperpolarization-gated PX, QP
HCN2 Hyperpolarization-gated PX, QP, IWQ
HCN3 Hyperpolarization-gated  
HCN4 Hyperpolarization-gated MP, PX, QP, IWQ
ICRAC Calcium release activated current PX
IK (KCa3.1) Potassium, calcium-activated PX, QP
Kir1.1 Potassium, inward rectifier  
Kir2.1 (IK1) Potassium, inward rectifier MP, PX, QP, IWQ
Kir3.1/Kir3.2 Potassium, inward rectifier  
Kir3.1/Kir3.4 Potassium, inward rectifier MP, PX
Kir6.1/SUR2B Potassium, inward rectifier PX
Kir6.2/SUR1 Potassium, inward rectifier PX
Kir6.2/SUR2A Potassium, inward rectifier MP, PX, FLP
Kir6.2/SUR2B Potassium, inward rectifier  
Kv1.1 Potassium, voltage-gated PX, QP
Kv1.2 Potassium, voltage-gated PX, QP, IWQ
Kv1.3 Potassium, voltage-gated PX, QP, IWQ
Kv1.4 Potassium, voltage-gated PX, QP, IWQ
Kv1.5 Potassium, voltage-gated MP, PX, QP, IWQ
Kv1.6 Potassium, voltage-gated  
Kv1.7 Potassium, voltage-gated  
Kv11.1 (hERG) Potassium, voltage-gated MP, PX, QP, IWQ
Kv2.1/Kv9.3 Potassium, voltage-gated  
Kv3.4 Potassium, voltage-gated PX, QP, IWQ
Kv4.1 Potassium, voltage-gated  
Kv4.2/KChIP2.2 Potassium, voltage-gated MP, PX, QP, IWQ
Kv4.3 Potassium, voltage-gated MP, PX, QP, IWQ
Kv4.3/KChIP2.2 Potassium, voltage-gated PX, QP
Kv7.1 (KCNQ1/KCNE2) Potassium, voltage-gated  
Kv7.1 (KvLQT1-minK; KCNQ1-KCNE1) Potassium, voltage-gated MP, PX, QP, IWQ, FLP
Kv7.2/Kv7.3 (KCNQ2/KCNQ3) Potassium, voltage-gated MP, PX, FLP
Kv7.2/Kv7.4 (KCNQ2/KCNQ4) Potassium, voltage-gated PX, QP, FLP
Kv7.3/Kv7.5 (KCNQ3/KCNQ5) Potassium, voltage-gated MP, PX, FLP
Kv7.4 (KCNQ4) Potassium, voltage-gated MP, PX, QP, FLP
MDR1 Multidrug resistance transporter FLP
Nav1.1 Sodium, voltage-gated MP, PX, QP, IWQ
Nav1.2 Sodium, voltage-gated MP, PX, QP, IWQ
Nav1.3 Sodium, voltage-gated MP, PX, QP, IWQ
Nav1.4 Sodium, voltage-gated PX, QP, IWQ
Nav1.5 Sodium, voltage-gated MP, PX, QP, IWQ
Nav1.6 Sodium, voltage-gated MP, PX, QP, IWQ
Nav1.7 Sodium, voltage-gated MP, PX, QP, IWQ, FLP
Nav1.8/β3 Sodium, voltage-gated PX, QP, IWQ
NCX1 Sodium/calcium exchanger MP, FLP
Nicotinic receptor (nAChR) α1 Ligand-gated PX
Nicotinic receptor (nAChR) α3 Ligand-gated PX
Nicotinic receptor (nAChR) α3/β4 Ligand-gated QP
Nicotinic receptor (nAChR) α4/β2 Ligand-gated  
Nicotinic receptor (nAChR) α7 Ligand-gated QP, FLP
NMDA receptor Ligand-gated PX
NMDA receptor (NR1/NR2A) Ligand-gated MP, FLP
NMDA receptor (NR1/NR2B) Ligand-gated MP, FLP
P2X1 Purinergic receptors MP, PX, FLP
P2X2 Purinergic receptors PX, FLP
P2X2/P2X3 Purinergic receptors PX, FLP
P2X3 Purinergic receptors MP, PX, FLP
P2X4 Purinergic receptors PX, FLP
P2X7 Purinergic receptors PX, QP, FLP
SK1 (KCa2.1) Potassium, calcium-activated QP
SK2 (KCa2.2) Potassium, calcium-activated QP, FLP
SK3 (KCa2.3) Potassium, calcium-activated MP, QP, FLP
TRPA1 TRP (transient receptor potential) MP, QP, FLP
TRPC1 TRP (transient receptor potential) MP
TRPC4 TRP (transient receptor potential) MP
TRPC6 TRP (transient receptor potential) MP, FLP
TRPM2 TRP (transient receptor potential) MP
TRPM4 TRP (transient receptor potential) MP, FLP
TRPM5 TRP (transient receptor potential)  
TRPM7 TRP (transient receptor potential)  
TRPM8 TRP (transient receptor potential) QP, FLP
TRPP1/TRPP2 TRP (transient receptor potential)  
TRPV1 TRP (transient receptor potential) MP, PX, FLP
TRPV2 TRP (transient receptor potential)  
TRPV4 TRP (transient receptor potential) MP, FLP
TRPV6 TRP (transient receptor potential) MP, PX

 

Download: Ion Channel targets and current platform validation list.

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